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Crystal structure of pre-activated arrestin p44

Yong Ju Kim, Klaus Peter Hofmann, Oliver P. Ernst, Patrick Scheerer (), Hui-Woog Choe () and Martha E. Sommer ()
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Yong Ju Kim: Institut für Medizinische Physik und Biophysik (CC2), Charité-Universitätsmedizin Berlin, Charitéplatz 1, D-10117 Berlin, Germany
Klaus Peter Hofmann: Institut für Medizinische Physik und Biophysik (CC2), Charité-Universitätsmedizin Berlin, Charitéplatz 1, D-10117 Berlin, Germany
Oliver P. Ernst: University of Toronto, 1 King’s College Circle
Patrick Scheerer: Institut für Medizinische Physik und Biophysik (CC2), AG Protein X-ray Crystallography, Charité-Universitätsmedizin Berlin, Charitéplatz 1, D-10117 Berlin, Germany
Hui-Woog Choe: Institut für Medizinische Physik und Biophysik (CC2), Charité-Universitätsmedizin Berlin, Charitéplatz 1, D-10117 Berlin, Germany
Martha E. Sommer: Institut für Medizinische Physik und Biophysik (CC2), Charité-Universitätsmedizin Berlin, Charitéplatz 1, D-10117 Berlin, Germany

Nature, 2013, vol. 497, issue 7447, 142-146

Abstract: The crystal structure of arrestin-1 is reported, in which the activation step is mimicked by C-tail truncation; the structure of this pre-activated arrestin is markedly different from the basal state and gives an insight into the activation mechanism.

Date: 2013
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DOI: 10.1038/nature12133

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