Intracellular allosteric antagonism of the CCR9 receptor

Christine Oswald, Mathieu Rappas, James Kean, Andrew S. Doré, James C. Errey, Kirstie Bennett, Francesca Deflorian, John A. Christopher, Ali Jazayeri, Jonathan S. Mason, Miles Congreve, Robert M. Cooke and Fiona H. Marshall ()
Additional contact information
Christine Oswald: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Mathieu Rappas: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
James Kean: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Andrew S. Doré: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
James C. Errey: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Kirstie Bennett: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Francesca Deflorian: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
John A. Christopher: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Ali Jazayeri: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Jonathan S. Mason: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Miles Congreve: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Robert M. Cooke: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City
Fiona H. Marshall: Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City

Nature, 2016, vol. 540, issue 7633, 462-465

Abstract: The crystal structure of the CCR9 chemokine receptor in complex with vercirnon at 2.8 Å resolution.

Date: 2016
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DOI: 10.1038/nature20606

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